Kajbaf, Mahmud

A comparative study of the CYP450 inhibition potential of marketed drugs using two fluorescence based assay platforms routinely used in the pharmaceutical industry. [electronic resource] - Drug metabolism letters Jan 2011 - 30-9 p. digital

Publication Type: Comparative Study; Journal Article

1874-0758

10.2174/187231211794455262 doi


Automation
Cell Line
Cytochrome P-450 Enzyme Inhibitors
Cytochrome P-450 Enzyme System--genetics
Dose-Response Relationship, Drug
Drug Discovery--methods
Drug Interactions
Enzyme Inhibitors--pharmacology
Escherichia coli--enzymology
Fluorescence
High-Throughput Screening Assays--methods
Humans
Microsomes--drug effects
Molecular Probes
Recombinant Proteins--antagonists & inhibitors
Reproducibility of Results
Substrate Specificity
Technology, Pharmaceutical--methods
Transfection