Bajjuri, Krishna Mohan

The legumain protease-activated auristatin prodrugs suppress tumor growth and metastasis without toxicity. [electronic resource] - ChemMedChem Jan 2011 - 54-9 p. digital

Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, U.S. Gov't, Non-P.H.S.

1860-7187

10.1002/cmdc.201000478 doi


Aminobenzoates--administration & dosage
Animals
Breast Neoplasms--drug therapy
Cell Line, Tumor
Cysteine Endopeptidases--metabolism
Disease Models, Animal
Enzyme Activation--drug effects
Female
Humans
Mice
Neoplasm Metastasis--drug therapy
Oligopeptides--administration & dosage
Prodrugs--administration & dosage
Tumor Burden--drug effects
Weight Loss--drug effects