Beck, Hilary P

Improvement of the synthesis and pharmacokinetic properties of chromenotriazolopyrimidine MDM2-p53 protein-protein inhibitors. [electronic resource] - Bioorganic & medicinal chemistry letters May 2011 - 2752-5 p. digital

Publication Type: Journal Article

1464-3405

10.1016/j.bmcl.2010.11.027 doi


Animals
Drug Stability
Humans
Infusion Pumps
Inhibitory Concentration 50
Molecular Structure
Proto-Oncogene Proteins c-mdm2--antagonists & inhibitors
Pyrimidines--chemical synthesis
Rats
Solubility
Structure-Activity Relationship
Tumor Suppressor Protein p53--antagonists & inhibitors