Superfamily-wide portrait of serine hydrolase inhibition achieved by library-versus-library screening. [electronic resource]
- Proceedings of the National Academy of Sciences of the United States of America Dec 2010
- 20941-6 p. digital
Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't
1091-6490
10.1073/pnas.1011663107 doi
Carbamates--pharmacology Catalytic Domain Drug Discovery--methods Drug Evaluation, Preclinical Enzyme Inhibitors--chemistry Fluorides Humans Hydrolases--antagonists & inhibitors Molecular Probes Phosphates Protein Binding Proteome Serine Small Molecule Libraries--pharmacology Substrate Specificity