Bachovchin, Daniel A

Superfamily-wide portrait of serine hydrolase inhibition achieved by library-versus-library screening. [electronic resource] - Proceedings of the National Academy of Sciences of the United States of America Dec 2010 - 20941-6 p. digital

Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't

1091-6490

10.1073/pnas.1011663107 doi


Carbamates--pharmacology
Catalytic Domain
Drug Discovery--methods
Drug Evaluation, Preclinical
Enzyme Inhibitors--chemistry
Fluorides
Humans
Hydrolases--antagonists & inhibitors
Molecular Probes
Phosphates
Protein Binding
Proteome
Serine
Small Molecule Libraries--pharmacology
Substrate Specificity