TY - GEN AU - Leslie,Colin P AU - Biagetti,Matteo AU - Bison,Silvia AU - Bromidge,Steven M AU - Di Fabio,Romano AU - Donati,Daniele AU - Falchi,Alessandro AU - Garnier,Martine J AU - Jaxa-Chamiec,Albert AU - Manchee,Gary AU - Merlo,Giancarlo AU - Pizzi,Domenica A AU - Stasi,Luigi P AU - Tibasco,Jessica AU - Vong,Antonio AU - Ward,Simon E AU - Zonzini,Laura TI - Discovery of 1-(3-{2-[4-(2-methyl-5-quinolinyl)-1-piperazinyl]ethyl}phenyl)-2-imidazolidinone (GSK163090), a Potent, selective, and orally active 5-HT1A/B/D receptor antagonist SN - 1520-4804 PY - 2014///0415 KW - Administration, Oral KW - Animals KW - CHO Cells KW - Chromatography, Liquid KW - Cricetulus KW - Drug Discovery KW - Humans KW - Imidazoles KW - administration & dosage KW - Magnetic Resonance Spectroscopy KW - Male KW - Quinolines KW - Rats, Sprague-Dawley KW - Receptors, Serotonin KW - classification KW - Serotonin Antagonists KW - Tandem Mass Spectrometry N1 - Publication Type: Journal Article UR - https://doi.org/10.1021/jm100714c ER -