Finley, Michael F A

An integrated multiassay approach to the discovery of small-molecule N-type voltage-gated calcium channel antagonists. [electronic resource] - Assay and drug development technologies Dec 2010 - 685-94 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1557-8127

10.1089/adt.2010.0311 doi


Analgesics--pharmacology
Animals
Calcitonin Gene-Related Peptide--metabolism
Calcium Channel Blockers--pharmacology
Calcium Channels, N-Type--metabolism
Cell Line
Ganglia, Spinal--metabolism
HEK293 Cells
High-Throughput Screening Assays
Humans
Luminescent Measurements
Neurons--metabolism
Pain--physiopathology
Patch-Clamp Techniques
Presynaptic Terminals--physiology
Rats
Small Molecule Libraries
Spinal Cord--metabolism
omega-Conotoxins--pharmacology