TY  - GEN
AU  - Kretzer,Nicole M
AU  - Cherian,Milu T
AU  - Mao,Chengjian
AU  - Aninye,Irene O
AU  - Reynolds,Philip D
AU  - Schiff,Rachel
AU  - Hergenrother,Paul J
AU  - Nordeen,Steven K
AU  - Wilson,Elizabeth M
AU  - Shapiro,David J
TI  - A noncompetitive small molecule inhibitor of estrogen-regulated gene expression and breast cancer cell growth that enhances proteasome-dependent degradation of estrogen receptor {alpha}
SN  - 1083-351X
PY  - 2011///0209
KW  - Breast Neoplasms
KW  - metabolism
KW  - Butyrophenones
KW  - chemistry
KW  - Cell Line, Tumor
KW  - Estrogen Receptor alpha
KW  - antagonists & inhibitors
KW  - Female
KW  - Fluorescence Polarization
KW  - Gene Expression Regulation, Neoplastic
KW  - Genes, Reporter
KW  - Humans
KW  - Leupeptins
KW  - pharmacology
KW  - Models, Chemical
KW  - Mucin-1
KW  - Proteasome Endopeptidase Complex
KW  - Purines
KW  - RNA, Messenger
KW  - Response Elements
KW  - Tamoxifen
KW  - analogs & derivatives
N1  - Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't
UR  - https://doi.org/10.1074/jbc.M110.183723
ER  -