TY - GEN AU - Symons,Kent T AU - Nguyen,Phan M AU - Massari,Mark E AU - Anzola,John V AU - Staszewski,Lena M AU - Wang,Li AU - Yazdani,Nahid AU - Dorow,Steven AU - Muhammad,Jerry AU - Sablad,Marciano AU - Rozenkrants,Natasha AU - Bonefous,Celine AU - Payne,Joseph E AU - Rix,Peter J AU - Shiau,Andrew K AU - Noble,Stewart A AU - Smith,Nicholas D AU - Hassig,Christian A AU - Zhang,Yan AU - Rao,Tadimeti S TI - Pharmacological characterization of KLYP961, a dual inhibitor of inducible and neuronal nitric-oxide synthases SN - 1521-0103 PY - 2011///0303 KW - Analgesics KW - pharmacology KW - Animals KW - Anti-Inflammatory Agents KW - Cells, Cultured KW - Cytochrome P-450 Enzyme Inhibitors KW - Enzyme Inhibitors KW - pharmacokinetics KW - Fluoroquinolones KW - Gastrointestinal Transit KW - drug effects KW - Humans KW - Macaca mulatta KW - Male KW - Mice KW - Mice, Inbred BALB C KW - Mice, Inbred C57BL KW - Motor Activity KW - Nitric Oxide Synthase Type I KW - antagonists & inhibitors KW - Nitric Oxide Synthase Type II KW - Protein Multimerization KW - Pyrazines N1 - Publication Type: Journal Article UR - https://doi.org/10.1124/jpet.110.172817 ER -