Symons, Kent T

Pharmacological characterization of KLYP961, a dual inhibitor of inducible and neuronal nitric-oxide synthases. [electronic resource] - The Journal of pharmacology and experimental therapeutics Feb 2011 - 468-78 p. digital

Publication Type: Journal Article

1521-0103

10.1124/jpet.110.172817 doi


Analgesics--pharmacology
Animals
Anti-Inflammatory Agents--pharmacology
Cells, Cultured
Cytochrome P-450 Enzyme Inhibitors
Enzyme Inhibitors--pharmacokinetics
Fluoroquinolones--pharmacokinetics
Gastrointestinal Transit--drug effects
Humans
Macaca mulatta
Male
Mice
Mice, Inbred BALB C
Mice, Inbred C57BL
Motor Activity--drug effects
Nitric Oxide Synthase Type I--antagonists & inhibitors
Nitric Oxide Synthase Type II--antagonists & inhibitors
Protein Multimerization
Pyrazines--pharmacokinetics