Tomasi, Sophie

Targeting the polyamine transport system with benzazepine- and azepine-polyamine conjugates. [electronic resource] - Journal of medicinal chemistry Nov 2010 - 7647-63 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1520-4804

10.1021/jm1007648 doi


Animals
Antineoplastic Agents--chemical synthesis
Azepines--chemical synthesis
Benzazepines--chemical synthesis
Biological Transport--drug effects
CHO Cells
Cell Proliferation--drug effects
Cricetinae
Cricetulus
Drug Screening Assays, Antitumor
Leukemia L1210
Polyamines--chemical synthesis
Spermidine--analogs & derivatives
Spermine--analogs & derivatives
Structure-Activity Relationship