Able, S L Receptor localization, native tissue binding and ex vivo occupancy for centrally penetrant P2X7 antagonists in the rat. [electronic resource] - British journal of pharmacology Jan 2011 - 405-14 p. digital Publication Type: Journal Article ISSN: 1476-5381 Standard No.: 10.1111/j.1476-5381.2010.01025.x doi Subjects--Topical Terms: AnimalsAutoradiographyBinding, CompetitiveBrain--metabolismCerebral Cortex--metabolismDrug DiscoveryGuanidines--bloodMaleMolecular Targeted TherapyProtein BindingPurinergic P2X Receptor Antagonists--metabolismQuinolines--bloodRadioligand AssayRatsRats, Sprague-DawleyReceptors, Purinergic P2X7--metabolismSpinal Cord--metabolism