Bettini, Ezio Identification and characterization of novel NMDA receptor antagonists selective for NR2A- over NR2B-containing receptors. [electronic resource] - The Journal of pharmacology and experimental therapeutics Dec 2010 - 636-44 p. digital Publication Type: Journal Article ISSN: 1521-0103 Standard No.: 10.1124/jpet.110.172544 doi Subjects--Topical Terms: AnimalsBinding, CompetitiveCalcium Signaling--drug effectsCell Line, TumorCell Membrane--metabolismCerebral Cortex--cytologyDrug Evaluation, Preclinical--methodsExcitatory Amino Acid Antagonists--chemistryExcitatory Postsynaptic Potentials--drug effectsFluorometry--methodsGlutamic Acid--pharmacologyGlycine--pharmacologyHEK293 CellsHumansMaleMolecular StructureN-Methylaspartate--pharmacologyNeurons--cytologyPatch-Clamp TechniquesRatsRats, Sprague-DawleyReceptors, N-Methyl-D-Aspartate--antagonists & inhibitorsTransfection