Bettini, Ezio

Identification and characterization of novel NMDA receptor antagonists selective for NR2A- over NR2B-containing receptors. [electronic resource] - The Journal of pharmacology and experimental therapeutics Dec 2010 - 636-44 p. digital

Publication Type: Journal Article

1521-0103

10.1124/jpet.110.172544 doi


Animals
Binding, Competitive
Calcium Signaling--drug effects
Cell Line, Tumor
Cell Membrane--metabolism
Cerebral Cortex--cytology
Drug Evaluation, Preclinical--methods
Excitatory Amino Acid Antagonists--chemistry
Excitatory Postsynaptic Potentials--drug effects
Fluorometry--methods
Glutamic Acid--pharmacology
Glycine--pharmacology
HEK293 Cells
Humans
Male
Molecular Structure
N-Methylaspartate--pharmacology
Neurons--cytology
Patch-Clamp Techniques
Rats
Rats, Sprague-Dawley
Receptors, N-Methyl-D-Aspartate--antagonists & inhibitors
Transfection