Rulcova, A

Stereoselective interactions of warfarin enantiomers with the pregnane X nuclear receptor in gene regulation of major drug-metabolizing cytochrome P450 enzymes. [electronic resource] - Journal of thrombosis and haemostasis : JTH Dec 2010 - 2708-17 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1538-7836

10.1111/j.1538-7836.2010.04036.x doi


Anticoagulants--chemistry
Cell Line, Tumor
Cytochrome P-450 Enzyme System--genetics
Fluorescence Resonance Energy Transfer
Gene Expression Regulation, Enzymologic--drug effects
Genes, Reporter
Humans
Pregnane X Receptor
Receptors, Steroid--drug effects
Reverse Transcriptase Polymerase Chain Reaction
Stereoisomerism
Transcriptional Activation
Two-Hybrid System Techniques
Up-Regulation--drug effects
Warfarin--chemistry