Bavisotto, Linda M

Tecarfarin, a novel vitamin K reductase antagonist, is not affected by CYP2C9 and CYP3A4 inhibition following concomitant administration of fluconazole in healthy participants. [electronic resource] - Journal of clinical pharmacology Apr 2011 - 561-74 p. digital

Publication Type: Journal Article; Randomized Controlled Trial; Research Support, Non-U.S. Gov't

1552-4604

10.1177/0091270010370588 doi


Administration, Oral
Adult
Aryl Hydrocarbon Hydroxylases--antagonists & inhibitors
Benzoates--administration & dosage
Coumarins--administration & dosage
Cytochrome P-450 CYP2C9
Cytochrome P-450 CYP3A
Cytochrome P-450 CYP3A Inhibitors
Drug Interactions
Enzyme Inhibitors--pharmacology
Female
Fluconazole--pharmacology
Humans
Male
NAD(P)H Dehydrogenase (Quinone)--antagonists & inhibitors
Warfarin--administration & dosage