Felts, Andrew S <br/><br/>
3-Cyano-5-fluoro-N-arylbenzamides as negative allosteric modulators of mGlu(5): Identification of easily prepared tool compounds with CNS exposure in rats.  [electronic resource] 

 -  Bioorganic & medicinal chemistry letters  Aug 2010 
 - 4390-4 p.  digital 
<br/><br/> Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't 
<br/><br/><label>ISSN: </label>1464-3405 
<br/><br/><label>Standard No.: </label>10.1016/j.bmcl.2010.06.064  doi 
<br/><br/><label>Subjects--Topical Terms: </label><br/>Allosteric Regulation<br/>Animals<br/>Benzamides--chemical synthesis<br/>Blood Proteins--metabolism<br/>Brain--metabolism<br/>Microsomes, Liver--metabolism<br/>Protein Binding<br/>Rats<br/>Receptor, Metabotropic Glutamate 5<br/>Receptors, Metabotropic Glutamate--antagonists & inhibitors<br/>Structure-Activity Relationship