Baffert, Fabienne
Potent and selective inhibition of polycythemia by the quinoxaline JAK2 inhibitor NVP-BSK805. [electronic resource]
- Molecular cancer therapeutics Jul 2010
- 1945-55 p. digital
Publication Type: Journal Article
ISSN: 1538-8514
Standard No.: 10.1158/1535-7163.MCT-10-0053 doi
Subjects--Topical Terms: Adenosine Triphosphate--pharmacology Animals Apoptosis--drug effects Cell Line Cell Line, Tumor Cell Proliferation--drug effects Erythropoiesis--drug effects Humans Janus Kinase 2--antagonists & inhibitors K562 Cells Mice Mice, Inbred BALB C Mice, SCID Models, Molecular Molecular Structure Mutation Phosphorylation--drug effects Polycythemia--metabolism Protein Structure, Tertiary Quinoxalines--chemistry Rats STAT5 Transcription Factor--metabolism Splenomegaly--metabolism