Docking of protein kinase B inhibitors: implications in the structure-based optimization of a novel scaffold. [electronic resource]
- Chemical biology & drug design Sep 2010
- 269-76 p. digital
Publication Type: Letter; Research Support, Non-U.S. Gov't
1747-0285
10.1111/j.1747-0285.2010.01002.x doi
Antineoplastic Agents--chemistry Crystallography, X-Ray Drug Discovery Models, Molecular Protein Kinase Inhibitors--chemistry Protein Structure, Tertiary Proto-Oncogene Proteins c-akt--antagonists & inhibitors Structure-Activity Relationship