Analogs of zanamivir with modified C4-substituents as the inhibitors against the group-1 neuraminidases of influenza viruses. [electronic resource]
- Bioorganic & medicinal chemistry Jun 2010
- 4074-84 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1464-3391
10.1016/j.bmc.2010.04.010 doi
Antiviral Agents--chemistry Enzyme Inhibitors--chemistry Influenza A Virus, H1N1 Subtype Inhibitory Concentration 50 Neuraminidase--antagonists & inhibitors Orthomyxoviridae--enzymology Protein Binding Protein Conformation Structure-Activity Relationship Zanamivir--analogs & derivatives