Organic cation transporters modulate the uptake and cytotoxicity of picoplatin, a third-generation platinum analogue. [electronic resource]
- Molecular cancer therapeutics Apr 2010
- 1058-69 p. digital
Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't
1538-8514
10.1158/1535-7163.MCT-09-1084 doi
Animals Cell Death--drug effects Cell Line, Tumor Cimetidine--pharmacology DNA Adducts--metabolism Gene Expression Regulation, Neoplastic--drug effects Humans Lung Neoplasms--genetics Mice Organic Cation Transport Proteins--antagonists & inhibitors Platinum Compounds--pharmacokinetics Polymorphism, Single Nucleotide--genetics Tissue Distribution--drug effects Xenograft Model Antitumor Assays