Zuercher, William J Discovery of tertiary sulfonamides as potent liver X receptor antagonists. [electronic resource] - Journal of medicinal chemistry Apr 2010 - 3412-6 p. digital Publication Type: Journal Article; Research Support, Non-U.S. Gov't ISSN: 1520-4804 Standard No.: 10.1021/jm901797p doi Subjects--Topical Terms: AnimalsCell LineCrystallography, X-RayHaplorhiniHumansLiver X ReceptorsModels, MolecularOrphan Nuclear Receptors--antagonists & inhibitorsStructure-Activity RelationshipSulfonamides--chemical synthesisTranscriptional Activation--drug effects