Zuercher, William J

Discovery of tertiary sulfonamides as potent liver X receptor antagonists. [electronic resource] - Journal of medicinal chemistry Apr 2010 - 3412-6 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1520-4804

10.1021/jm901797p doi


Animals
Cell Line
Crystallography, X-Ray
Haplorhini
Humans
Liver X Receptors
Models, Molecular
Orphan Nuclear Receptors--antagonists & inhibitors
Structure-Activity Relationship
Sulfonamides--chemical synthesis
Transcriptional Activation--drug effects