Bursavich, Matthew G

Novel benzofuran-3-one indole inhibitors of PI3 kinase-alpha and the mammalian target of rapamycin: hit to lead studies. [electronic resource] - Bioorganic & medicinal chemistry letters Apr 2010 - 2586-90 p. digital

Publication Type: Journal Article

1464-3405

10.1016/j.bmcl.2010.02.082 doi


Benzofurans--chemistry
Cell Line, Tumor
Humans
Intracellular Signaling Peptides and Proteins--antagonists & inhibitors
Models, Molecular
Phosphoinositide-3 Kinase Inhibitors
Protein Kinase Inhibitors--chemistry
Protein Serine-Threonine Kinases--antagonists & inhibitors
Structure-Activity Relationship
TOR Serine-Threonine Kinases