Novel benzofuran-3-one indole inhibitors of PI3 kinase-alpha and the mammalian target of rapamycin: hit to lead studies. [electronic resource]
- Bioorganic & medicinal chemistry letters Apr 2010
- 2586-90 p. digital
Publication Type: Journal Article
1464-3405
10.1016/j.bmcl.2010.02.082 doi
Benzofurans--chemistry Cell Line, Tumor Humans Intracellular Signaling Peptides and Proteins--antagonists & inhibitors Models, Molecular Phosphoinositide-3 Kinase Inhibitors Protein Kinase Inhibitors--chemistry Protein Serine-Threonine Kinases--antagonists & inhibitors Structure-Activity Relationship TOR Serine-Threonine Kinases