Mutations that increase both Hsp90 ATPase activity in vitro and Hsp90 drug resistance in vivo. [electronic resource]
- Biochimica et biophysica acta May 2010
- 575-83 p. digital
Publication Type: Journal Article
0006-3002
10.1016/j.bbamcr.2010.03.002 doi
Adenosine Triphosphatases--metabolism Amino Acid Substitution Benzoquinones--pharmacology Blotting, Western Chaperonins--genetics Drug Resistance Enzyme Inhibitors--pharmacology HSP90 Heat-Shock Proteins--antagonists & inhibitors Humans Immunoprecipitation In Vitro Techniques Kidney--embryology Lactams, Macrocyclic--pharmacology Models, Molecular Molecular Chaperones--genetics Mutation--genetics Protein Binding Protein Conformation Saccharomyces cerevisiae--genetics Saccharomyces cerevisiae Proteins--genetics Two-Hybrid System Techniques