Rajapakse, Hemaka A SAR of tertiary carbinamine derived BACE1 inhibitors: role of aspartate ligand amine pKa in enzyme inhibition. [electronic resource] - Bioorganic & medicinal chemistry letters Mar 2010 - 1885-9 p. digital Publication Type: Journal Article ISSN: 1464-3405 Standard No.: 10.1016/j.bmcl.2010.01.137 doi Subjects--Topical Terms: Amines--metabolismAmyloid Precursor Protein Secretases--antagonists & inhibitorsAspartic Acid--metabolismAspartic Acid Endopeptidases--antagonists & inhibitorsCatalysisEnzyme Inhibitors--pharmacologyHumansModels, MolecularStructure-Activity Relationship