Mechanistic characterization and molecular modeling of hepatitis B virus polymerase resistance to entecavir. [electronic resource]
- PloS one Feb 2010
- e9195 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1932-6203
10.1371/journal.pone.0009195 doi
Amino Acid Sequence Amino Acid Substitution Antiviral Agents--pharmacology Binding Sites--genetics Drug Resistance, Viral--genetics Guanine--analogs & derivatives Guanosine Triphosphate--chemistry Hep G2 Cells Hepatitis B virus--enzymology Humans Hydrogen Bonding Kinetics Lamivudine--pharmacology Models, Molecular Protein Binding Protein Structure, Tertiary RNA-Directed DNA Polymerase--chemistry Substrate Specificity Viral Proteins--chemistry Virus Replication--drug effects