3-Aryl-4-(arylhydrazono)-1H-pyrazol-5-ones: Highly ligand efficient and potent inhibitors of GSK3beta. [electronic resource]
- Bioorganic & medicinal chemistry letters Mar 2010
- 1661-4 p. digital
Publication Type: Journal Article
1464-3405
10.1016/j.bmcl.2010.01.072 doi
Binding Sites Crystallography, X-Ray Glycogen Synthase Kinase 3--antagonists & inhibitors Glycogen Synthase Kinase 3 beta Ligands Protein Binding Protein Kinase Inhibitors--chemical synthesis Protein Kinases--chemistry Pyrazolones--chemical synthesis Structure-Activity Relationship