TY  - GEN
AU  - Rose,Nathan R
AU  - Woon,Esther C Y
AU  - Kingham,Guy L
AU  - King,Oliver N F
AU  - Mecinović,Jasmin
AU  - Clifton,Ian J
AU  - Ng,Stanley S
AU  - Talib-Hardy,Jobina
AU  - Oppermann,Udo
AU  - McDonough,Michael A
AU  - Schofield,Christopher J
TI  - Selective inhibitors of the JMJD2 histone demethylases: combined nondenaturing mass spectrometric screening and crystallographic approaches
SN  - 1520-4804
PY  - 2010///0323
KW  - Binding Sites
KW  - Binding, Competitive
KW  - Combinatorial Chemistry Techniques
KW  - Crystallography, X-Ray
KW  - Humans
KW  - Jumonji Domain-Containing Histone Demethylases
KW  - antagonists & inhibitors
KW  - Models, Molecular
KW  - Oxalates
KW  - chemical synthesis
KW  - Spectrometry, Mass, Electrospray Ionization
KW  - Spectrometry, Mass, Matrix-Assisted Laser Desorption-Ionization
KW  - Structure-Activity Relationship
KW  - Tyrosine
KW  - analogs & derivatives
N1  - Publication Type: Journal Article; Research Support, Non-U.S. Gov't
UR  - https://doi.org/10.1021/jm901680b
ER  -