Rose, Nathan R

Selective inhibitors of the JMJD2 histone demethylases: combined nondenaturing mass spectrometric screening and crystallographic approaches. [electronic resource] - Journal of medicinal chemistry Feb 2010 - 1810-8 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1520-4804

10.1021/jm901680b doi


Binding Sites
Binding, Competitive
Combinatorial Chemistry Techniques
Crystallography, X-Ray
Humans
Jumonji Domain-Containing Histone Demethylases--antagonists & inhibitors
Models, Molecular
Oxalates--chemical synthesis
Spectrometry, Mass, Electrospray Ionization
Spectrometry, Mass, Matrix-Assisted Laser Desorption-Ionization
Structure-Activity Relationship
Tyrosine--analogs & derivatives