Activation of the cystic fibrosis transmembrane conductance regulator by the flavonoid quercetin: potential use as a biomarker of ΔF508 cystic fibrosis transmembrane conductance regulator rescue. [electronic resource]
- American journal of respiratory cell and molecular biology Nov 2010
- 607-16 p. digital
Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't
1535-4989
10.1165/rcmb.2009-0281OC doi
Animals Biomarkers--metabolism Cell Membrane--drug effects Chlorides--metabolism Cyclic AMP--metabolism Cystic Fibrosis Transmembrane Conductance Regulator--chemistry Dose-Response Relationship, Drug Drug Evaluation, Preclinical Humans Ion Channel Gating--drug effects Ion Transport--drug effects Membrane Potentials--drug effects Mice Mutant Proteins--chemistry NIH 3T3 Cells Nasal Mucosa--drug effects Phosphorylation--drug effects Protein Structure, Tertiary Quercetin--pharmacology Rats Receptors, Adrenergic, beta-2--metabolism