Pyle, Louise C

Activation of the cystic fibrosis transmembrane conductance regulator by the flavonoid quercetin: potential use as a biomarker of ΔF508 cystic fibrosis transmembrane conductance regulator rescue. [electronic resource] - American journal of respiratory cell and molecular biology Nov 2010 - 607-16 p. digital

Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't

1535-4989

10.1165/rcmb.2009-0281OC doi


Animals
Biomarkers--metabolism
Cell Membrane--drug effects
Chlorides--metabolism
Cyclic AMP--metabolism
Cystic Fibrosis Transmembrane Conductance Regulator--chemistry
Dose-Response Relationship, Drug
Drug Evaluation, Preclinical
Humans
Ion Channel Gating--drug effects
Ion Transport--drug effects
Membrane Potentials--drug effects
Mice
Mutant Proteins--chemistry
NIH 3T3 Cells
Nasal Mucosa--drug effects
Phosphorylation--drug effects
Protein Structure, Tertiary
Quercetin--pharmacology
Rats
Receptors, Adrenergic, beta-2--metabolism