Rilatt, Ian
Discovery and SAR of small molecule PAR1 antagonists. [electronic resource]
- Bioorganic & medicinal chemistry letters Feb 2010
- 903-6 p. digital
Publication Type: Comparative Study; Journal Article
1464-3405
10.1016/j.bmcl.2009.12.072 doi
Animals
CHO Cells
Cricetinae
Cricetulus
Drug Discovery--methods
Humans
Microsomes, Liver--drug effects
Oligopeptides--chemistry
Protease Inhibitors--chemistry
Rats
Receptor, PAR-1--physiology
Structure-Activity Relationship
Platelet Aggregation Inhibitors