Rilatt, Ian

Discovery and SAR of small molecule PAR1 antagonists. [electronic resource] - Bioorganic & medicinal chemistry letters Feb 2010 - 903-6 p. digital

Publication Type: Comparative Study; Journal Article

1464-3405

10.1016/j.bmcl.2009.12.072 doi


Animals
CHO Cells
Cricetinae
Cricetulus
Drug Discovery--methods
Humans
Microsomes, Liver--drug effects
Oligopeptides--chemistry
Protease Inhibitors--chemistry
Rats
Receptor, PAR-1--physiology
Structure-Activity Relationship
Platelet Aggregation Inhibitors