TY - GEN AU - Kawasaki,Yuko AU - Chufan,Eduardo E AU - Lafont,Virginie AU - Hidaka,Koushi AU - Kiso,Yoshiaki AU - Mario Amzel,L AU - Freire,Ernesto TI - How much binding affinity can be gained by filling a cavity? SN - 1747-0285 PY - 2010///0330 KW - Binding Sites KW - Calorimetry KW - Crystallography, X-Ray KW - Drug Design KW - HIV Protease Inhibitors KW - chemistry KW - Humans KW - Hydrogen Bonding KW - Protein Binding KW - Protein Structure, Tertiary KW - Thermodynamics N1 - Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't UR - https://doi.org/10.1111/j.1747-0285.2009.00921.x ER -