How much binding affinity can be gained by filling a cavity? [electronic resource]
- Chemical biology & drug design Feb 2010
- 143-51 p. digital
Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't
1747-0285
10.1111/j.1747-0285.2009.00921.x doi
Binding Sites Calorimetry Crystallography, X-Ray Drug Design HIV Protease Inhibitors--chemistry Humans Hydrogen Bonding Protein Binding Protein Structure, Tertiary Thermodynamics