Yu, Weiping

Synthesis, radiolabeling, and biological evaluation of (R)- and (S)-2-amino-3-[(18)F]fluoro-2-methylpropanoic acid (FAMP) and (R)- and (S)-3-[(18)F]fluoro-2-methyl-2-N-(methylamino)propanoic acid (NMeFAMP) as potential PET radioligands for imaging brain tumors. [electronic resource] - Journal of medicinal chemistry Jan 2010 - 876-86 p. digital

Publication Type: Journal Article; Research Support, N.I.H., Extramural

1520-4804

10.1021/jm900556s doi


Amino Acids--pharmacokinetics
Aminoisobutyric Acids--chemical synthesis
Animals
Biological Transport
Brain Neoplasms--diagnosis
Cell Line, Tumor
Isotope Labeling--methods
Positron-Emission Tomography--methods
Radiopharmaceuticals--chemical synthesis
Rats
Tissue Distribution