Ahmad, Saleem

Tricyclic dihydroquinazolinones as novel 5-HT2C selective and orally efficacious anti-obesity agents. [electronic resource] - Bioorganic & medicinal chemistry letters Feb 2010 - 1128-33 p. digital

Publication Type: Comparative Study; Journal Article; Research Support, Non-U.S. Gov't

1464-3405

10.1016/j.bmcl.2009.12.014 doi


Administration, Oral
Animals
Anti-Obesity Agents--administration & dosage
Eating--drug effects
Humans
Male
Obesity--drug therapy
Protein Binding--physiology
Quinazolinones--administration & dosage
Rats
Rats, Sprague-Dawley
Receptor, Serotonin, 5-HT2C--metabolism
Serotonin 5-HT2 Receptor Agonists
Serotonin Receptor Agonists--administration & dosage