Langsdorf, Erik F

Screening for antibacterial inhibitors of the UDP-3-O-(R-3-hydroxymyristoyl)-N-acetylglucosamine deacetylase (LpxC) using a high-throughput mass spectrometry assay. [electronic resource] - Journal of biomolecular screening Jan 2010 - 52-61 p. digital

Publication Type: Journal Article

1552-454X

10.1177/1087057109355319 doi


Amidohydrolases--antagonists & inhibitors
Anti-Bacterial Agents--analysis
Dimethyl Sulfoxide--pharmacology
Enzyme Inhibitors--analysis
Enzyme Stability--drug effects
Escherichia coli--drug effects
Fluorescence
High-Throughput Screening Assays--methods
Mass Spectrometry--methods
Microbial Sensitivity Tests
Reproducibility of Results
Small Molecule Libraries--analysis
Substrate Specificity--drug effects
Temperature