Screening for antibacterial inhibitors of the UDP-3-O-(R-3-hydroxymyristoyl)-N-acetylglucosamine deacetylase (LpxC) using a high-throughput mass spectrometry assay. [electronic resource]
- Journal of biomolecular screening Jan 2010
- 52-61 p. digital
Publication Type: Journal Article
1552-454X
10.1177/1087057109355319 doi
Amidohydrolases--antagonists & inhibitors Anti-Bacterial Agents--analysis Dimethyl Sulfoxide--pharmacology Enzyme Inhibitors--analysis Enzyme Stability--drug effects Escherichia coli--drug effects Fluorescence High-Throughput Screening Assays--methods Mass Spectrometry--methods Microbial Sensitivity Tests Reproducibility of Results Small Molecule Libraries--analysis Substrate Specificity--drug effects Temperature