Kumar, Sanjeev Metabolism and excretion of anacetrapib, a novel inhibitor of the cholesteryl ester transfer protein, in humans. [electronic resource] - Drug metabolism and disposition: the biological fate of chemicals Mar 2010 - 474-83 p. digital Publication Type: Clinical Trial; Comparative Study; Journal Article ISSN: 1521-009X Standard No.: 10.1124/dmd.109.028704 doi Subjects--Topical Terms: AdolescentAdultAnticholesteremic Agents--adverse effectsBiotransformationCholesterol Ester Transfer Proteins--antagonists & inhibitorsCytochrome P-450 CYP3A--geneticsCytochrome P-450 CYP3A InhibitorsCytochrome P-450 Enzyme InhibitorsCytochrome P-450 Enzyme System--geneticsFeces--chemistryHumansIsoenzymes--antagonists & inhibitorsMaleMicrosomes, Liver--enzymologyMiddle AgedMolecular StructureOxazolidinones--adverse effectsRecombinant Proteins--antagonists & inhibitorsTandem Mass SpectrometryYoung Adult