Novel and selective DNA methyltransferase inhibitors: Docking-based virtual screening and experimental evaluation. [electronic resource]
- Bioorganic & medicinal chemistry Jan 2010
- 822-9 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1464-3391
10.1016/j.bmc.2009.11.050 doi
Cloning, Molecular Crystallography, X-Ray DNA (Cytosine-5-)-Methyltransferase 1 DNA (Cytosine-5-)-Methyltransferases--antagonists & inhibitors Dose-Response Relationship, Drug Drug Evaluation, Preclinical Enzyme Inhibitors--chemistry Humans Models, Molecular Structure-Activity Relationship DNA Methyltransferase 3B