Blakemore, David C
Synthesis and in vivo evaluation of bicyclic gababutins. [electronic resource]
- Bioorganic & medicinal chemistry letters Jan 2010
- 461-4 p. digital
Publication Type: Journal Article
1464-3405
10.1016/j.bmcl.2009.11.118 doi
Amines--chemical synthesis
Amino Acids--chemical synthesis
Animals
Blood-Brain Barrier--metabolism
Bridged Bicyclo Compounds--chemical synthesis
CHO Cells
Cricetinae
Cricetulus
Cyclohexanecarboxylic Acids--chemical synthesis
Gabapentin
Neuralgia--drug therapy
Pain Measurement
Rats
Stereoisomerism
Structure-Activity Relationship
gamma-Aminobutyric Acid--chemical synthesis