TY - GEN AU - Sabbatini,Fabio M AU - Di Fabio,Romano AU - Griffante,Cristiana AU - Pentassuglia,Giorgio AU - Zonzini,Laura AU - Melotto,Sergio AU - Alvaro,Giuseppe AU - Capelli,Anna M AU - Pippo,Lara AU - Perdona',Elisabetta AU - St Denis,Yves AU - Costa,Silvano AU - Corsi,Mauro TI - Synthesis and pharmacological characterization of constrained analogues of Vestipitant as in vitro potent and orally active NK(1) receptor antagonists SN - 1464-3405 PY - 2010///0420 KW - Anti-Anxiety Agents KW - chemical synthesis KW - Drug Design KW - Fluorobenzenes KW - Humans KW - Molecular Conformation KW - Neurokinin-1 Receptor Antagonists KW - Piperidines KW - Receptors, Neurokinin-1 KW - metabolism N1 - Publication Type: Journal Article UR - https://doi.org/10.1016/j.bmcl.2009.11.078 ER -