Sabbatini, Fabio M <br/><br/>
Synthesis and pharmacological characterization of constrained analogues of Vestipitant as in vitro potent and orally active NK(1) receptor antagonists.  [electronic resource] 

 -  Bioorganic & medicinal chemistry letters  Jan 2010 
 - 623-7 p.  digital 
<br/><br/> Publication Type: Journal Article 
<br/><br/><label>ISSN: </label>1464-3405 
<br/><br/><label>Standard No.: </label>10.1016/j.bmcl.2009.11.078  doi 
<br/><br/><label>Subjects--Topical Terms: </label><br/>Anti-Anxiety Agents--chemical synthesis<br/>Drug Design<br/>Fluorobenzenes<br/>Humans<br/>Molecular Conformation<br/>Neurokinin-1 Receptor Antagonists<br/>Piperidines--chemical synthesis<br/>Receptors, Neurokinin-1--metabolism