TY  - GEN
AU  - Sally,Elliott J
AU  - Xu,Heng
AU  - Dersch,Christina M
AU  - Hsin,Ling-Wei
AU  - Chang,Li-Te
AU  - Prisinzano,Thomas E
AU  - Simpson,Denise S
AU  - Giuvelis,Denise
AU  - Rice,Kenner C
AU  - Jacobson,Arthur E
AU  - Cheng,Kejun
AU  - Bilsky,Edward J
AU  - Rothman,Richard B
TI  - Identification of a novel "almost neutral" micro-opioid receptor antagonist in CHO cells expressing the cloned human mu-opioid receptor
SN  - 1098-2396
PY  - 2010///0510
KW  - Analgesics, Opioid
KW  - pharmacology
KW  - Animals
KW  - CHO Cells
KW  - drug effects
KW  - Cricetinae
KW  - Cricetulus
KW  - Dose-Response Relationship, Drug
KW  - Furans
KW  - Gene Expression Regulation
KW  - Guanosine 5'-O-(3-Thiotriphosphate)
KW  - metabolism
KW  - Humans
KW  - Narcotic Antagonists
KW  - chemistry
KW  - Protein Binding
KW  - Pyrones
KW  - Receptors, Opioid, mu
KW  - antagonists & inhibitors
KW  - Sulfur Isotopes
N1  - Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, N.I.H., Intramural
UR  - https://doi.org/10.1002/syn.20723
ER  -