Distinct pose of discodermolide in taxol binding pocket drives a complementary mode of microtubule stabilization. [electronic resource]
- Biochemistry Dec 2009
- 11664-77 p. digital
Publication Type: Comparative Study; Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't
1520-4995
10.1021/bi901351q doi
Alkanes--chemistry Animals Binding Sites--drug effects Carbamates--chemistry Cattle Chickens Deuterium Exchange Measurement Dimerization Drug Synergism Lactones--chemistry Microtubules--chemistry Paclitaxel--chemistry Peptide Fragments--blood Protein Binding--drug effects Protein Isoforms--blood Protein Stability--drug effects Pyrones--chemistry Tubulin--blood Tubulin Modulators--chemistry