Trova, Michael P

Heterobiaryl purine derivatives as potent antiproliferative agents: inhibitors of cyclin dependent kinases. Part II. [electronic resource] - Bioorganic & medicinal chemistry letters Dec 2009 - 6613-7 p. digital

Publication Type: Journal Article

1464-3405

10.1016/j.bmcl.2009.10.011 doi


Antineoplastic Agents--chemical synthesis
Cell Proliferation--drug effects
Cyclin-Dependent Kinases--antagonists & inhibitors
Drug Design
Drug Screening Assays, Antitumor
HeLa Cells
Humans
Molecular Structure
Protein Kinase Inhibitors--chemical synthesis
Purines--chemical synthesis
Roscovitine
Stereoisomerism
Structure-Activity Relationship