Glucuronidation and covalent protein binding of benoxaprofen and flunoxaprofen in sandwich-cultured rat and human hepatocytes. [electronic resource]
- Drug metabolism and disposition: the biological fate of chemicals Dec 2009
- 2314-22 p. digital
Publication Type: Comparative Study; Journal Article; Research Support, N.I.H., Extramural
1521-009X
10.1124/dmd.109.028944 doi
Adult Animals Anti-Inflammatory Agents, Non-Steroidal--metabolism Benzoxazoles--metabolism Biotransformation Cell Culture Techniques Collagen Dose-Response Relationship, Drug Drug Combinations Feasibility Studies Glucuronates--metabolism Glucuronosyltransferase--metabolism Hepatocytes--metabolism Humans Ibuprofen--metabolism Kinetics Laminin Male Microsomes, Liver--metabolism Models, Biological Propionates--metabolism Protein Binding Proteoglycans Rats Rats, Sprague-Dawley