TY - GEN AU - Mowbray,Charles E AU - Burt,Catherine AU - Corbau,Romuald AU - Gayton,Simon AU - Hawes,Michael AU - Perros,Manos AU - Tran,Isabelle AU - Price,David A AU - Quinton,Faye J AU - Selby,Matthew D AU - Stupple,Paul A AU - Webster,Rob AU - Wood,Anthony TI - Pyrazole NNRTIs 4: selection of UK-453,061 (lersivirine) as a development candidate SN - 1464-3405 PY - 2010///0105 KW - Acquired Immunodeficiency Syndrome KW - drug therapy KW - Animals KW - Anti-HIV Agents KW - chemical synthesis KW - Cell Line KW - Drug Resistance, Viral KW - HIV Reverse Transcriptase KW - antagonists & inhibitors KW - Humans KW - Microsomes, Liver KW - metabolism KW - Nitriles KW - Pyrazoles KW - Rats KW - Reverse Transcriptase Inhibitors N1 - Publication Type: Journal Article UR - https://doi.org/10.1016/j.bmcl.2009.08.080 ER -