C-5 Substituted heteroaryl 3-pyridinecarbonitriles as PKCtheta inhibitors: Part I. [electronic resource]
- Bioorganic & medicinal chemistry letters Sep 2009
- 5423-5 p. digital
Publication Type: Journal Article
1464-3405
10.1016/j.bmcl.2009.07.109 doi
Animals Inhibitory Concentration 50 Isoenzymes--antagonists & inhibitors Mice Mice, Knockout Nitriles--chemistry Protein Kinase C--antagonists & inhibitors Protein Kinase C-theta Protein Kinase Inhibitors--chemistry Pyridines--chemistry Structure-Activity Relationship T-Lymphocytes--drug effects