Aubry, Carine

Fascaplysin-inspired diindolyls as selective inhibitors of CDK4/cyclin D1. [electronic resource] - Bioorganic & medicinal chemistry Aug 2009 - 6073-84 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1464-3391

10.1016/j.bmc.2009.06.070 doi


Binding Sites
Computer Simulation
Cyclin A--antagonists & inhibitors
Cyclin D1--antagonists & inhibitors
Cyclin-Dependent Kinase 2--antagonists & inhibitors
Cyclin-Dependent Kinase 4--antagonists & inhibitors
Drug Design
Humans
Indoles--chemical synthesis
Protein Kinase Inhibitors--chemical synthesis