Castagnolo, Daniele

Synthesis, biological evaluation, and SAR study of novel pyrazole analogues as inhibitors of Mycobacterium tuberculosis: part 2. Synthesis of rigid pyrazolones. [electronic resource] - Bioorganic & medicinal chemistry Aug 2009 - 5716-21 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1464-3391

10.1016/j.bmc.2009.05.058 doi


Animals
Antitubercular Agents--chemical synthesis
Chlorocebus aethiops
Computer Simulation
Microbial Sensitivity Tests
Models, Molecular
Mycobacterium tuberculosis--drug effects
Pyrazolones--chemical synthesis
Structure-Activity Relationship
Tuberculosis--drug therapy
Vero Cells