Blood-brain barrier transport of naloxone does not involve P-glycoprotein-mediated efflux. [electronic resource]
- Journal of pharmaceutical sciences Jan 2010
- 413-21 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1520-6017
10.1002/jps.21819 doi
ATP Binding Cassette Transporter, Subfamily B ATP Binding Cassette Transporter, Subfamily B, Member 1--antagonists & inhibitors Animals Biological Transport Blood-Brain Barrier--metabolism Brain--metabolism Dose-Response Relationship, Drug Half-Life HeLa Cells Humans In Vitro Techniques Male Microinjections Models, Biological Naloxone--administration & dosage Narcotic Antagonists--administration & dosage Rats Rats, Wistar Tissue Distribution