Kazi, Aslamuzzaman

Discovery of a novel proteasome inhibitor selective for cancer cells over non-transformed cells. [electronic resource] - Cell cycle (Georgetown, Tex.) Jun 2009 - 1940-51 p. digital

Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't

1551-4005

10.4161/cc.8.12.8798 doi


Animals
Anthracyclines--chemistry
Antineoplastic Agents--chemistry
Boronic Acids--chemistry
Bortezomib
Cell Line, Tumor
Cell Proliferation--drug effects
Cell Survival--drug effects
Chymotrypsin--antagonists & inhibitors
Cyclin-Dependent Kinase Inhibitor p27
Drug Discovery
Humans
Inhibitory Concentration 50
Intracellular Signaling Peptides and Proteins--agonists
Mice
Mice, Nude
Neoplasms--enzymology
Proteasome Inhibitors
Protein Conformation
Pyrazines--chemistry
Serine Proteinase Inhibitors--chemistry
Small Molecule Libraries
Xenograft Model Antitumor Assays