Strakhova, M I

In vitro and in vivo characterization of A-940894: a potent histamine H4 receptor antagonist with anti-inflammatory properties. [electronic resource] - British journal of pharmacology May 2009 - 44-54 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1476-5381

10.1111/j.1476-5381.2009.00236.x doi


Animals
Anti-Inflammatory Agents, Non-Steroidal--pharmacokinetics
Binding, Competitive
Calcium--metabolism
Cell Shape
Chemotaxis
Eosinophils--drug effects
Female
Histamine--pharmacology
Humans
Male
Mast Cells--cytology
Mice
Mice, Inbred BALB C
Peritonitis--chemically induced
Piperazines--pharmacokinetics
Prostaglandin D2--metabolism
Pyrimidines--pharmacokinetics
RNA, Messenger--biosynthesis
Radioligand Assay
Rats
Rats, Sprague-Dawley
Receptors, G-Protein-Coupled--antagonists & inhibitors
Receptors, Histamine--biosynthesis
Receptors, Histamine H4
Recombinant Proteins--antagonists & inhibitors
Zymosan